купить 99.8% Ингибитор ароматазы чистоты AI Форместан (Lentaron) порошок Интернет
What is Formestane?
Форместан – один из лучших легальных антиэстрогенов., и он классифицируется как необратимый ингибитор арроматазы., значение, разрушает фермент ароматазу.
Форместан представляет собой синтетическое стероидное вещество с противоопухолевой активностью, необратимо связывается с ферментом ароматазы и ингибирует его., thereby blocking the conversion of cholesterol to pregnenolone and the peripheral aromatization of androgenic precursors into estrogens. Formestane is a drug that has been previously used in breast cancer treatment. Like most drugs which have some sort of phsyique usage, athletes eventually get a hold of it.
Formestane Certificate Of Analysis
наименование товара |
Форместан |
Производственная баня |
20190108 |
Дата производства |
2019-01-08 |
Спецификация |
Стандарт предприятия |
Срок годности |
2 лет |
Количество |
100кг |
Дата анализа |
2019-01-08 |
|
|
|
|
Результат для анализа |
Предметы |
стандарт |
Результаты |
Тестовое задание |
Спецификация |
Результаты |
Внешность |
Белый или почти белый кристаллический порошок |
Удовлетворяет |
Температура плавления |
199-203℃ |
201.5℃ |
Убыток от высыхания |
0.50% |
0.32% |
Удельное вращение |
+172~+182° |
+174.5 ~+181° |
анализ |
not less than 97% |
99.8% |
Заключение |
Conforms Specifications of Enterprise Standard. |
Formestane Benefits:
1) Increases in IGF-1
2) Lowers SHBG to make anabolic hormones more active and in a free state
3) Increase natural Testosterone to above normal human levels and continues to work even after use has stopped.
4) Lowers and Controls Estrogen and prevents the negative side effects associated with Estrogen
5) Prevents Estrogen Rebound because it is a Type I aromatase Inhibitor similar to Aromasin (Exemestanes)
6) Prevents conversion of Testosterone to DHT meaning it can help prevent hair loss in some cases as well as prostate issues.
7) Transdermal Delivery allows for maximum absorption with zero toxicity and mess
Formestane Dosage:
Formestane Sufficient dosage of 200-400mg per day.
Formestane Active life 24-36 часов, usually last you about 3-4 недель.
Some evidence to suggest that higher response rates are achieved with Formestane/Lentaron 500 versus 250mg once every 2 недель. The clinical efficacy of intramuscular formestane 250mg did not differ significantly from that of oral megestrol when administered as second-line endocrine therapy to patients with advanced disease in whom previous tamoxifen therapy had failed.
К тому же, Formestane/Lentaron produced a response rate, duration of response and overall survival rate that was not significantly different from that of oral tamoxifen when administered as first-line endocrine therapy to patients with advanced disease, but tamoxifen was superior in some measures.
Formestane Chemical Profile
кличка |
Lentaron, 4-hydroxyandrost-4-ene-3,17-dione |
CAS НЕТ. |
566-48-3 |
Внешность |
off-white crystalline powder |
M Ж |
C19H26O3 |
M Вт |
302.41 |
Применение |
antitumor drug. aromatase inhibitor |
Оценка |
Фармацевтический класс |
дозировка |
250мг, 1 time every two weeks, as the arm deep intramuscular injection. |
плотность |
1.19 г / см3 |
Температура плавления |
199-202℃ |
Точка кипения |
475.4 в 760 мм рт.ст. |
Точка возгорания |
255.4 |